基本信息
分子式 | C32H31N3O5 |
分子量 | 537.61 |
MDL编码 | MFCD00132118 |
存储条件 | Freezer -20℃ |
半岛bd体育手机客户端 描述
KT5720 is a cell-permeable, potent, specific, reversible, ATP-competitive inhibitor of protein kinase A (PKA), with a Ki of 60 nM[1][2].
靶点(IC50 & Targe)
Ki: 60 nM (PKA)[1][2].
参考文献
[1]. Davies SP, et al. Specificity and mechanism of action of some commonly used protein kinase inhibitors. Biochem J. 2000 Oct 1;351(Pt 1):95-105.
[2]. Murray A, et al. Pharmacological PKA inhibition: all may not be what it seems. Sci Signal. 2008 Jun 3;1(22):re4.
安全信息
防范说明 | P262 |
WGK | 3 |
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