LY2033298

半岛bd体育手机客户端 说明

包装

5, 25 mg in glass bottle

生化/生理作用

LY2033298 is a robust allosteric potentiator that is highly selective for the human M4 muscarinic acetylcholine receptor subtype. LY2033298 potentiates ACh-M4 binding, with no effect at M1/3/5 receptors. LY2033298 can also bind to the M ACh receptor, and mediate either positive or negative allosteric effects depending on the ligand used to probe receptor activity.

特点和优势

This compound was developed by Eli Lilly. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

基本信息

经验(实验)分子式	C13H14ClN3O2S
分子量	311.79
MDL编号	MFCD12912423
PubChem化学物质编号	329817677
NACRES	NA.77

半岛bd体育手机客户端 性质

质量水平	100
测定	≥98% (HPLC)
形式	solid
储存条件	desiccated
颜色	off-white to tan
溶解性	DMSO: >20 mg/mL
创始人	Eli Lilly
储存温度	?20℃
SMILES string	COc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl
InChI	1S/C13H14ClN3O2S/c1-5-7-9(15)10(11(18)16-6-3-4-6)20-13(7)17-12(19-2)8(5)14/h6H,3-4,15H2,1-2H3,(H,16,18)
InChI key	CTEGQKDJTBWFHW-UHFFFAOYSA-N

安全信息

象形图
警示用语：	Danger
危险声明	H334
预防措施声明	P261 - P284 - P501
危险分类	Resp. Sens. 1
储存分类代码	11 - Combustible Solids
WGK	WGK 3
闪点(F)	Not applicable
闪点(C)	Not applicable