包装: | 5mg |
生物活性 |
[Ala1,3,11,15]-Endothelin (53-63) (TFA) is anETBagonist. [Ala1,3,11,15]-Endothelin (53-63) (TFA) has selectivity for ETBwithIC50values range from 0.33 nM to 0.61 nM. [Ala1,3,11,15]-Endothelin (53-63) (TFA) can be used for the research of vasoconstriction[1][2]. |
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IC50& Target[1] |
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体外研究 (In Vitro) |
[Ala1,3,11,15]-Endothelin (53-63) (TFA) (0.1 μM) has selectivity for ETBwith IC50values of 0.61 nM, 0.61 nM, 0.33 nM, 2200 nM in Bronchus, Lung, Cerebellum and VSMC, respectively[1].
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分子量 |
2481.70 |
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Formula |
C111H164F3N25O34S |
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Sequence |
Ala-Ser-Ala-Ser-Ser-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp |
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Sequence Shortening |
ASASSLMDKEAVYFAHLDIIW |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |