L-798,106 是一种有效且高度选择性的前列腺素 EP3 受体拮抗剂 (Ki\u003d0.3 nM),它还对 EP4、EP1 和 EP2 受体具有微摩尔活性,Ki 值分别为 916 nM、\u003e5000 nM 和 \u003e5000 nM。
Cas No. |
244101-02-8 |
别名 |
CM9; GW671021 |
化学名 |
(Z)-N-((5-bromo-2-methoxyphenyl)sulfonyl)-3-(2-(naphthalen-2-ylmethyl)phenyl)acrylamide |
Canonical SMILES |
BrC1=CC=C(C(S(=O)(NC(/C=C\C2=CC=CC=C2CC3=CC=C4C(C=CC=C4)=C3)=O)=O)=C1)OC |
分子式 |
C27H22BrNO4S |
分子量 |
536.44 |
溶解度 |
DMF: 20 mg/ml,DMSO: 10 mg/ml |
储存条件 |
Store at -20°C |
General tips |
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition |
Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |