CAS: |
204067-01-6 |
分子式: |
C32H36N6O5 |
分子量: |
584.67 |
纯度: |
>98% |
溶解性: |
DMSO |
存储: |
Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months; -20℃ 1 month |
研究领域: |
Cancer |
Target: |
Ki: 0.17 nM (Human BB1 receptor), 0.66 nM (Rat BB1 receptor), 1 nM (Human BB2 receptor), 16 nM (Rat BB2 receptor)[1];EC50: 0.31 μM (FPR1), 0.66 μM (FPR2)[2] |
描述: |
PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 n |