SDZ-216525 is a 5-HT1A receptor antagonist which significantly inhibits the tracheal contractions induced both by NKA (10 nM-3 microM) and 5-HT (10 nM-10 microM) (n=4-10). References: Germonpré PR, Joos GF, Pauwels RA. Modulation by 5-HT1A receptors of the 5-HT2 receptor-mediated tachykinin-induced contraction of the rat trachea in vitro. Br J Pharmacol. 1998 Apr;123(8):1571-8. PubMed PMID: 9605563; PubMed Central PMCID: PMC1565327.
纯度:≥98%
CAS:141533-35-9