RU 24969 hemisuccinate 是一种优先的 5-HT1B 激动剂,Ki 为 0.38 nM,但对 5-HT1A 受体 (Ki=2.5 nM) 也显示出明显的亲和力,并且对大脑中的其他受体位点具有低亲和力。
货号:ajcx26756
CAS:66611-27-6
分子式:C14H16N2O.?C4H6O4
分子量:287.34
溶解度:DMF: slightly soluble,DMSO: slightly soluble,Ethanol: slightly soluble,PBS (pH 7.2): 1 mg/ml
纯度:98%
存储:Store at -20°C
库存:
现货
Background:
Potent 5-HT1A/1B and moderate 5-HT2C agonist that may also release 5-HT. Centrally active following systemic administration.
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