Glutaminase-IN-3 (compound 657) 是一种有效的 glutaminase 抑制剂，对GLS1的 IC50 值为0.24 μM。详细情况请参见专利 WO2014089048A1，compound 657。
货号:ajcx33420
CAS:1439399-45-7
分子式:C19H19F3N6O2S
分子量：452.45
溶解度:DMSO : 50 mg/mL (110.51 mM; Need ultrasonic)
纯度：98%
存储：Store at -20°C
库存： 现货

Background:

Glutaminase-IN-3 (compound 657) is a potent glutaminase inhibitor with an IC50 of 0.24 μM for Glutaminase 1 (GLS1). Glutaminase-IN-3 is extracted from patent WO2014089048A1, compound 657[1].

[1]. Mark K. Bennett, et al. Treatment of cancer with heterocyclic inhibitors of glutaminase. WO2014089048A1.