LG-100064是一种类视黄醇X受体(retinoid-X-receptor(RXR))激动剂,对RXRα,RXRβ和RXRγ的EC50值分别为330nM,200nM和260nM;LG-100064可用于癌症研究。
货号:ajcx13138
CAS:153559-46-7
分子式:C23H26O3
分子量:350.45
溶解度:Soluble in DMSO
纯度:98%
存储:Store at -20°C
库存:
现货
Background:
LG-100064 is a retinoid-X-receptor (RXR) agonist, with EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ; LG-100064 can be used in the research of cancer.
LG-100064 (3-Methyl-TTNCB) is a retinoid-X-receptor (RXR) agonist, with EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ. LG-100064 shows no effect on RARα/β/γ (EC50, >10000 nM)[1].
[1]. Marcus F. Boehm, et al. Compounds having selective activity for retinoid X receptors, and means for modulation of processes mediated by retinoid X receptors.