FR252384是一种有效的neuropeptideY-Y5receptor拮抗剂,IC50值为2.3nM。
CAS:447405-11-0
分子式:C18H17N3
分子量:275.35
纯度:98%
存储:Store at -20°C
Background:
FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM.
FR252384 is orally absorbable and permeable to brain[1].
[1]. Satoh Y, et al. Novel potent antagonists of human neuropeptide Y-Y5 receptor. Part 4: tetrahydrodiazabenzazulene derivatives. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1009-11.