B-Raf IN 5 (化合物 3b) 是一种有效的蛋白激酶
B-Raf抑制剂,
IC50为 2.0 nM。B-Raf IN 5 不与二级靶点 PXR 结合,并能抵抗快速代谢。B-Raf IN 5 具有研究癌症疾病的潜力。
生物活性 |
B-Raf IN 5 (compound 3b) is a potent inhibitor of protein kinaseB-Rafwith anIC50of 2.0 nM. B-Raf IN 5 is devoid of binding to the secondary target PXR and resists rapid metabolism. B-Raf IN 6 has the potential for the research ofcancerdisease[1].
|
分子量 |
|
Formula |
|
CAS 号 |
|
运输条件 |
Room temperature in continental US; may vary elsewhere.
|
储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis.
|