AM8936 是一种平衡且有效的 1 型大麻素受体 (CB1) 激动剂（对 rCB1 和 hCB1 的
EC50分别为 8.6 和 1.4 nM)。AM8936 对 rCB1 具有高亲和力，
Ki为 0.55 nM。AM8936 在体内对 CB1 受体也具有激活作用。AM8936 可用于研究 CNS 和代谢紊乱、疼痛、青光眼等。
| 生物活性 |
AM8936 acts as a balanced and potentcannabinoid receptortype-1 (CB1) agonist in functional assays (EC50s of 8.6 and 1.4 nM for rCB1 and hCB1, respectively). AM8936 exhibits high affinity for ratCB1(rCB1) withKiof 0.55 nM. AM8936 is a potent and efficaciousCB1 agonistin vivo. AM8936 can be used for the research of CNS and metabolic disorders, pain, glaucoma, etc[1].
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis.
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