MNI137 是一种有效的选择性负变构调节剂,适用于 II 组 mGluR。MNI137 对人和大鼠 mGlu2 抑制谷氨酸诱导的钙动员的
IC50s值为 8.3 和 12.6 nM。
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MNI137 is a potent and selective negative allosteric modulator for group II mGluRs. MNI137 hasIC50svalues of 8.3 and 12.6 nM for human and rat mGlu2 inhibition of glutamate-induced calcium mobilization[1].
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运输条件 |
Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
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